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January 1, 2014

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Functionalised staple linkages for modulating the cellular activity of stapled peptides

YLYu Heng LauThe University of Sydney PAPeterson de AndradeUniversity of Manchester SQS.T. QuahAgency for Science, Technology and Research

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Resumen

A divergent synthetic strategy for generating helical p53 peptides bearing functionalised staple linkages, allowing for efficient optimisation of cellular activity.

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Cite This Study

Lau et al. (Wed,) studied this question.

synapsesocial.com/papers/69d852ba8c03fbaff8bef092 https://doi.org/https://doi.org/10.1039/c4sc00045e

Functionalised staple linkages for modulating the cellular activity of stapled peptides | Synapse

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