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Gem -difluorinated alkoxyphenyl group conformational and DMPK properties modulation experimentally demonstrated in a macrocyclic system.
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Thomas J. Cogswell
AstraZeneca (Netherlands)
Richard J. Lewis
AstraZeneca (Netherlands)
Christian Sköld
Uppsala University
Chemical Science
Uppsala University
AstraZeneca (Sweden)
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Cogswell et al. (Mon,) studied this question.
synapsesocial.com/papers/6a1acccb77ec05d9a7b8dc18 — DOI: https://doi.org/10.1039/d4sc05424e