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November 14, 2025PharmaceuticsOpen Access

Polyphenol-Rich Citrullus lanatus Rind Extract Mitigates Doxorubicin-Induced Cardiotoxicity: HPLC Profiling and In Vivo Evaluation

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Why the study?

Cardiovascular diseases remain a major global cause of mortality driven partly by oxidative stress and inflammation, prompting evaluation of the cardioprotective potential of polyphenol-rich Citrullus lanatus rind extract against doxorubicin-induced cardiotoxicity.

Does polyphenol-rich Citrullus lanatus rind extract mitigate doxorubicin-induced cardiotoxicity in rats?

Population

30 healthy male Wistar Kyoto rats

Comparison

PRCL extract at 250 or 500 mg/kg/day vs quercetin vs control in doxorubicin-treated rats

Design

In vivo randomized animal study with in vitro assay

Follow-up

21 days

Key result

Polyphenol-rich Citrullus lanatus rind extract (500 mg/kg/day) mitigated doxorubicin-induced cardiotoxicity in rats, restoring antioxidant biomarkers and reducing inflammatory cytokines.

Authors

BABader Alsuwayt

Discussion

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Overview

Should not yet change doxorubicin cardiotoxicity management; leaves open translation of rat findings to human trials.

Structured PICO

Does polyphenol-rich Citrullus lanatus rind extract mitigate doxorubicin-induced cardiotoxicity in rats?

P
Population
30 healthy male Wistar Kyoto rats treated with doxorubicin (10 mg/kg) to induce cardiotoxicity
I
Intervention
Polyphenol-rich Citrullus lanatus (PRCL) rind extract administered at 250 and 500 mg/kg/day for 21 days
C
Comparator
Standard quercetin group and doxorubicin-only control
O
Outcome
Cardiovascular markers, antioxidant biomarkers (SOD, CAT, GPx, GSH), lipid peroxidation (MDA), inflammatory cytokines (TNF-α, IL-6), and histopathological examination of cardiac tissuesurrogate

Polyphenol-rich Citrullus lanatus rind extract demonstrates antioxidant and cardioprotective properties against doxorubicin-induced cardiotoxicity in a rat model.

Cite This Study

Bader Alsuwayt (2025) studied Doxorubicin-induced cardiotoxicity (n=30). Polyphenol-rich Citrullus lanatus (PRCL) rind extract vs. Doxorubicin alone and standard quercetin was evaluated on Cardiovascular markers, antioxidant biomarkers, lipid peroxidation, and inflammatory cytokines. Polyphenol-rich Citrullus lanatus rind extract (500 mg/kg/day) mitigated doxorubicin-induced cardiotoxicity in rats, restoring antioxidant biomarkers and reducing inflammatory cytokines.

synapsesocial.com/papers/6a1c5dcb01af05bf0da93613https://doi.org/10.3390/pharmaceutics17111469
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