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October 2, 2025Organic Letters2 citations

Chemodivergent Synthesis of Multiborylalkanes via Deoxygenative Polyborylation of Silyl Enol Ethers

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WDWenke DongHMHonghui MaWZWanxiang Zhao

Key Points

  • Cobalt-catalyzed deoxygenative polyborylation yields multiple multiborylalkane types effectively.
  • The method allows synthesis of 1,1,1-triborylalkanes, 1,1,3-triborylalkanes, and 1,1-diborylalkenes.
  • Utilizing HBpin favors formation of 1,1-diborylalkanes under mild conditions and broad substrate scope.
  • Mechanistic investigations indicate processes initiated via dehydrogenative and deoxygenative borylation.

Abstract

A cobalt-catalyzed, chemodivergent deoxygenative polyborylation strategy for silyl enol ethers has been developed, enabling selective synthesis of 1,1,1-triborylalkanes, 1,1,3-triborylalkanes, 1,1-diborylalkenes, and 1,1-diborylalkanes. Specifically, deoxygenative borylation with B2pin2 affords 1,1,1-triborylalkanes, 1,1,3-triborylalkanes, and 1,1-diborylalkenes, while the use of HBpin favors 1,1-diborylalkane formation. This protocol offers mild reaction conditions, a broad substrate scope, and high functional group tolerance. The utility and practicality of this method were demonstrated through gram-scale reactions and various product transformations. Mechanistic investigations revealed that all processes are initiated via the cobalt-catalyzed dehydrogenative and deoxygenative borylation of silyl enol ethers.

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Cite This Study

Dong et al. (2025) studied this question.

synapsesocial.com/papers/68de79595b556a9128e1a180https://doi.org/10.1021/acs.orglett.5c03751
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