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December 8, 2025BloodOpen Access

Phase 3 randomized double-blind study evaluating selinexor, an XPO1 inhibitor, plus ruxolitinib in jaki-naïve myelofibrosis: Study rationale and preliminary patient characteristics

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Authors

SGSebastian GrosickiHAHaris AliLULaura Urian

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Overview

Phase 3 trial demonstrates safety and tolerability of selinexor with ruxolitinib in myelofibrosis, indicating potential for improved treatment outcomes.

Key Points

  • This study aims to evaluate the efficacy and safety of selinexor combined with ruxolitinib in patients with JAKi-naïve myelofibrosis.
  • Phase 3 randomized double-blind trial.
  • Participants receive selinexor and ruxolitinib versus placebo plus ruxolitinib.
  • Endpoints include safety, tolerability, progression-free survival, and pharmacokinetics.
  • Safety profile shows acceptable tolerability with reported adverse events including nausea and anemia.
  • Outcomes measured include SVR35 and Abs-TSS at week 24, with trials ongoing.
  • Analysis of health care resource utilization will be included in the final evaluation.

Cite This Study

Grosicki et al. (2025) studied this question.

synapsesocial.com/papers/69362f6e4fa91c937236e075https://doi.org/10.1182/blood-2025-7353
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