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March 14, 2026Organic & Biomolecular Chemistry2 citations

Glycosyl modified nucleoside motifs for glycoconjugation of oligonucleotides

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BMBiju MajumdarHAHaythem AbdaHBHenri Barry

Key Points

  • The aim is to create carbohydrate-oligonucleotide conjugates for specific receptor targeting.
  • Synthesis of glycosyl-nucleoside moieties linked to thymine via a 1,2,3-triazole linker
  • Utilization of click chemistry for bioconjugate preparation
  • Design of conjugates to engage specific sugar receptors
  • Successfully synthesized novel carbohydrate-oligonucleotide conjugates
  • Conjugates are designed to interact with glucose transporters and other sugar receptors
  • The method offers a reliable route for glycosylation of oligonucleotides

Abstract

The synthesis of novel carbohydrate-oligonucleotide conjugates is described. These bioconjugates, which feature glycosyl-nucleoside moieties linked to a thymine base via a 1,2,3-triazole linker, were prepared using a 'click' chemistry route. This synthetic approach enables the generation of oligonucleotide conjugates designed to engage specific sugar receptors, including glucose transporters as well as GalNAc and maltoheptaose-binding receptors.

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Cite This Study

Majumdar et al. (2026) studied this question.

synapsesocial.com/papers/69b4adc718185d8a39801b2dhttps://doi.org/10.1039/d5ob01901j
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