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April 15, 2026Advanced ScienceOpen Access

Antibody targeting integrin β3 β-tail suppresses platelet aggregation without inducing bleeding in preclinical models.

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Why the study?

Current antiplatelet drugs targeting integrin αIIbβ3 or its upstream signaling increase the risk of serious spontaneous bleeding, creating a need for safer antithrombotic strategies that prevent thrombosis without impairing normal hemostasis.

Does an antibody targeting the β-tail domain of integrin β3 prevent thrombosis without inducing bleeding in preclinical models?

Population

Ex vivo and in vivo models

Comparison

Antibody targeting the β-tail domain of integrin β3

Design

Preclinical experimental study

Key result

An antibody targeting the β-tail domain of integrin β3 suppressed platelet aggregation in ex vivo and in vivo models without inducing bleeding.

Authors

JLJoonha LeeCLChul-Gyun LimPVPothiappan Vairaprakash

Discussion

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Member takes

Overview

May enable antithrombotic benefit without bleeding risk; extends β-tail domain targeting of integrin β3 as selective therapeutic strategy.

Key Points

  • The aim is to create a safer method to prevent thrombosis without compromising normal blood clotting functions.
  • Targeted the beta-tail domain of integrin beta3 for antibody development.
  • The antibody selectively blocks force-induced activation of integrin alphaIIb beta3.
  • Evaluated efficacy in ex vivo and in vivo models.
  • The antibody successfully inhibits force-dependent alphaIIb beta3 activation.
  • Platelet aggregation at atherosclerotic lesions is significantly suppressed.
  • No spontaneous bleeding events were observed.

Structured PICO

Does an antibody targeting the β-tail domain of integrin β3 prevent thrombosis without inducing bleeding in preclinical models?

P
Population
ex vivo and in vivo models of platelet aggregation and thrombosis
I
Intervention
Antibody targeting the β-tail domain of integrin β3
O
Outcome
Platelet aggregation and bleeding risksurrogate

Targeting the β-tail domain of integrin β3 to selectively block force-induced activation provides a promising antithrombotic strategy that minimizes bleeding risk.

Cite This Study

Lee et al. (2026) studied Thrombosis. Antibody targeting the β-tail domain of integrin β3 was evaluated on Platelet aggregation and bleeding. An antibody targeting the β-tail domain of integrin β3 suppressed platelet aggregation in ex vivo and in vivo models without inducing bleeding.

synapsesocial.com/papers/69df2c1de4eeef8a2a6b11c3https://doi.org/10.1002/advs.202522086
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