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October 27, 1998CirculationOpen Access

BetaAR stimulation significantly increases the expression of betaARK1, whereas beta-blockade decreases expression.

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Why the study?

Does beta-adrenergic receptor stimulation or blockade alter the in vivo expression of betaARK1?

Population

In vivo model (specific model not detailed in abstract)

Design

Preclinical

Authors

GIGuido IaccarinoETEric D. TomhaveRLRobert J. Lefkowitz

Discussion

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Overview

May reduce betaARK1 to mediate beta-blocker benefits in HF; leaves open translation from animal models to humans.

Structured PICO

Does beta-adrenergic receptor stimulation or blockade alter the in vivo expression of betaARK1?

P
Population
In vivo model (specific model not detailed in abstract)
I
Intervention
Beta-adrenergic receptor (betaAR) stimulation and beta-blockade
O
Outcome
Myocardial G protein-coupled receptor kinase (betaARK1) expressionsurrogate

Demonstrates a novel mechanism of ligand-induced betaAR regulation where beta-blockade decreases betaARK1 expression, providing insight into the efficacy of beta-blockers in heart failure.

Cite This Study

Iaccarino et al. (1998) studied this question.

synapsesocial.com/papers/69eedef3a84321e0ae63c611https://doi.org/10.1161/01.cir.98.17.1783
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