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May 16, 2026Molecular and Cellular Biology0 citationsOpen Access

Pharmacological Inhibition of Valosin-Containing Protein (VCP) Triggers Cardiac Hypertrophy and Heart Failure in Vivo

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FDFederica DiofanoBABenedict AllhoffDPDeung-Dae Park

Key Points

  • This research investigates the effects of valosin-containing protein (VCP) inhibition on cardiac development and function.
  • Utilized zebrafish model to observe cardiac effects of VCP inhibition during different developmental stages (24-72 hpf and 72-120 hpf).
  • Assessed cardiac impairment, apoptosis, hypertrophy, and contractile function
  • Evaluated markers of proteostasis and endoplasmic reticulum (ER) stress.
  • Inhibition at early developmental stages caused severe cardiac impairment and increased apoptosis.
  • Inhibition during late stages led to ventricular hypertrophy with maintained contractile function.
  • VCP inhibition correlated with disrupted proteostasis and activation of ER stress, linking to cardomyopathy.

Abstract

knockout phenotypes. Early developmental inhibition (24-72 hpf) led to severe cardiac impairment and apoptosis, whereas inhibition during late development (72-120 hpf) induced ventricular hypertrophy with preserved contractile function, suggesting a developmental stage-dependent effect. Furthermore, Vcp inhibition was associated with markers of disrupted proteostasis, suggesting UPS dysfunction and ER stress activation. These findings establish a zebrafish model of VCP-related cardiomyopathy, highlight its role in cardiac proteostasis and hypertrophic remodeling, and provide novel insights into disease mechanisms and potential therapeutic targets.

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Cite This Study

Diofano et al. (2026) studied this question.

synapsesocial.com/papers/6a0808ffa487c87a6a40b20bhttps://doi.org/10.1080/10985549.2026.2664584
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