Population
Mice with cardiac-restricted overexpression of PPARalpha (MHC-PPAR)
Design
Preclinical
Key result
Cardiac-restricted overexpression of PPARα in mice increased myocardial fatty acid oxidation by 64% and decreased glucose oxidation by 63%, mimicking the metabolic phenotype of diabetic cardiomyopathy.
Authors
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Supports PPARα as mediator of diabetic cardiomyopathy-like metabolism; leaves open clinical relevance in humans.
Absolute Event Rate: 294% vs 179%
p-value: p=<0.05
Cardiac-restricted overexpression of PPARalpha in mice induces metabolic derangements and cardiomyopathy that mimic the diabetic heart, highlighting the maladaptive role of altered energy metabolism in diabetic cardiomyopathy.
Finck et al. (2002) studied Diabetic cardiomyopathy. Cardiac-restricted overexpression of PPARα vs. Nontransgenic littermates was evaluated on Myocardial palmitate oxidation rate (nmol/min/g dry weight) (p=<0.05). Cardiac-restricted overexpression of PPARα in mice increased myocardial fatty acid oxidation by 64% and decreased glucose oxidation by 63%, mimicking the metabolic phenotype of diabetic cardiomyopathy.