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April 6, 2023Open Access

The PLN R14del+/- mutation resulted in hyperdynamic Ca2+ handling, including a 43% reduction in Ca2+ transient decay kinetics, indicating a loss of SERCA2a inhibition rather than superinhibition.

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Why the study?

SERCA2a superinhibition is widely assumed to cause PLN-R14del-associated cardiomyopathy, but alternative mechanisms like abnormal energy metabolism are reported. This study evaluated Ca2+ dynamics and energy metabolism prior to cardiomyopathy development.

Population

Ventricular myocytes of 8-12 weeks-old, phenotypically silent, TG mice

Comparison

PLN R14del +/- mutation effects vs pharmacological PLN antagonism

Design

Preclinical transgenic mouse study

Key result

The PLN R14del+/- mutation resulted in hyperdynamic Ca2+ handling, including a 43% reduction in Ca2+ transient decay kinetics, indicating a loss of SERCA2a inhibition rather than superinhibition.

Authors

CMClaudia ManiezziMEMarem EskandrCFChiara Florindi

Discussion

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Overview

Challenges superinhibition hypothesis in young PLN R14del mice; leaves open ER stress or SR-mito uncoupling as early ACM drivers in patients.

Structured PICO

P
Population
Transgenic mice carrying the heterozygous phospholamban mutation R14del (PLN R14del+/-) aged 8 to 12 weeks, evaluated prior to the development of overt cardiomyopathy.
E
Exposure
Evaluation of the PLN R14del+/- mutation and pharmacological PLN antagonism with PST-3093.
C
Comparator
Wild-type (WT) littermates and untreated mutant cardiomyocytes.
O
Outcome
Ca2+ dynamics (including SERCA2a ATPase activity and intracellular Ca2+ transients) and energy metabolism parameters (oxygen consumption rate and proton efflux rate).surrogate

Main Result

Effect estimate: 43% reduction

Absolute Event Rate: 284% vs 495%

p-value: p=<0.0001

The PLN R14del+/- mutation causes hyperdynamic Ca2+ handling and depressed resting energy metabolism prior to cardiomyopathy development, challenging the prevailing SERCA2a superinhibition hypothesis.

Limitations

  • Because of technical constraints, metabolic measurements were performed in unstimulated (quiescent) cardiomyocytes.

Cite This Study

Maniezzi et al. (2023) studied Arrhythmogenic cardiomyopathy. PLN R14del+/- mutation vs. Wild-type (WT) littermates was evaluated on Ca2+ transient decay kinetics (τ decay) (43% reduction, p=<0.0001). The PLN R14del+/- mutation resulted in hyperdynamic Ca2+ handling, including a 43% reduction in Ca2+ transient decay kinetics, indicating a loss of SERCA2a inhibition rather than superinhibition.

synapsesocial.com/papers/6a7a108abdf697b3de027e07https://doi.org/10.1101/2023.04.05.535536
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