Copper efficiently catalyzed nucleophilic ring opening, sp 3 C–H functionalization, and C–N bond formation in the presence of tert -butyl hydroperoxide to afford functionalized imidazolidines starting from N -sulfonylaziridines and N -alkylanilines. The products were obtained in high optical purities (95 → 99% ee) with excellent functional group tolerance.
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Sengoden et al. (2016) studied this question.
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