Abstract 5‐Trifluoromethylthio‐substituted pyrimidines have been synthezised by halogenation of 5‐trifluoromethylthiouracile or barbituric acid with phosphorus halogenides POX3. The new compounds themselves are excellent starting materials for further nucleophilic exchange reactions. Thus fluoro‐, iodo‐, alkoxy‐ and aminoligands were introduced and further used for new synthesis. A new method for introducing trifluoromethylthio (SCF3)‐groups is presented.
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HAAS et al. (1986) studied this question.
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