Population
Pairs of neonatal rat heart cells
Comparison
Doxyl stearic acids (16-DSA and 12-DSA) vs Control conditions, methyl esters of 16- and…
Design
Preclinical
Key result
Doxyl stearic acids (16-DSA and 12-DSA) rapidly and reversibly reduced gap junctional conductance to unmeasurable levels in a dose- and time-dependent manner in neonatal rat heart cells.
Authors
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Supports hypothesis that ischemia-induced fatty acids promote arrhythmias via gap junction uncoupling; animal data leave mechanism unproven in vivo.
Doxyl stearic acids uncouple cardiac cells by reducing gap junctional conductance, suggesting a mechanism by which ischemia-induced free fatty acids may cause arrhythmias.
Janis M. Burt (1989) studied this question. Doxyl stearic acids (16-DSA and 12-DSA) vs. Methyl esters of 16- and 12-DSA, stearic acid, TEMPO, and control conditions was evaluated on Gap junctional conductance (gj). Doxyl stearic acids (16-DSA and 12-DSA) rapidly and reversibly reduced gap junctional conductance to unmeasurable levels in a dose- and time-dependent manner in neonatal rat heart cells.