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December 18, 2015Cell Death DiscoveryOpen Access

Selective cytoprotective effect of histamine on doxorubicin-induced hepatic and cardiac toxicity in animal models

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Key result

Histamine pretreatment prevents doxorubicin-induced cardiac damage and enhances anti-tumor activity in animal models.

Why the study?

The potential protective effect of histamine on doxorubicin-induced hepatic and cardiac toxicity required evaluation in rodent models and triple-negative breast cancer models.

Does histamine prevent doxorubicin-induced hepatic and cardiac toxicity in rodent models?

Population

Male Sprague Dawley rats, Balb/c mice, and human MDA-MB-231 triple-negative breast tumor-bearing mice

Comparison

Control vs histamine vs Dox vs Dox+histamine

Design

Preclinical animal and in vitro/in vivo laboratory study

Follow-up

2 weeks

Authors

MNM B NicoudHSHelena SterleECEliana Carabajal

Discussion

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Member takes

Overview

Does not support clinical use; leaves open translation of histamine cytoprotection from rodent doxorubicin models to patients.

Structured PICO

Does histamine prevent doxorubicin-induced hepatic and cardiac toxicity in rodent models?

P
Population
Preclinical animal study evaluating male Sprague Dawley rats, Balb/c mice, and female athymic nude mice treated with doxorubicin and histamine.
I
Intervention
Histamine (5 mg/kg for rats and 1 mg/kg for mice, daily subcutaneous injection starting 24 h before treatment) combined with doxorubicin (2 mg/kg, intraperitoneally injected three times a week for 2 weeks)
C
Comparator
Doxorubicin alone (2 mg/kg, intraperitoneally injected three times a week for 2 weeks), histamine alone, and control (saline)
O
Outcome
Tissue toxicity evaluated by histopathological studies, oxidative stress, and biochemical parameterssurrogate

Histamine demonstrates preclinical potential as a selective cytoprotective agent against doxorubicin-induced cardiotoxicity and hepatotoxicity without compromising anti-tumor efficacy.

Limitations

  • Preclinical animal model
  • Requires further studies to identify the specific histamine receptor subtype involved
  • Needs translation to clinical practice

Cite This Study

Nicoud et al. (2015) studied Doxorubicin-induced hepatic and cardiac toxicity. Histamine vs. Doxorubicin alone or saline was evaluated on Cardiac and hepatic tissue toxicity and tumor growth. Pretreatment with histamine prevented doxorubicin-induced cardiac and hepatic tissue damage by reducing oxidative stress and apoptosis, while preserving and enhancing the anti-tumor activity of doxorubicin in animal models.

synapsesocial.com/papers/6aa8016d871ca30df5b185c6https://doi.org/10.1038/cddiscovery.2015.59
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Also Consider

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  1. 1The histamine H4 receptor: from orphan to the clinic2015 · 138 citations
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  3. 3Histamine protects against the acute phase of experimentally-induced hepatic ischemia/re-perfusion2012 · 7 citations
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  5. 5Therapeutic potential of histamine <scp>H<sub>4</sub></scp> receptor agonists in triple‐negative human breast cancer experimental model2013 · 48 citations