Tandem reactions produced diastereomers through a one-pot synthesis under mild conditions, suggesting efficient pathways for complex compounds.
Copper‐catalyzed reactions of 2‐benzothiazolimines, terminal ynones, and sulfonyl azides afforded benzothiazolopyrimidine diastereomers. The transformation involved a tandem CuAAC/ring‐cleavage/[4 + 2] cycloaddition procedure with one‐pot synthesis under mild conditions. The benzothiazolopyrimidine diastereomers could be isolated, and their structure is confirmed by X‐ray single‐crystal diffraction.
No takes yet. Share an insight, caveat, or question.
Jing Shen (2025) studied this question.
Synapse has enriched 5 closely related papers on similar clinical questions. Consider them for comparative context: