Synapse
⌘+K
Synapse
PulseExploreClubsResearchersJournals
Instagram
HomeClubsExplore
January 11, 2018Drug Discovery TodayOpen Access

Progress with covalent small-molecule kinase inhibitors

View Full Paper
Ask AI
Bookmark
Share

Authors

ZZZheng ZhaoNanjing University of Chinese MedicinePBPhilip E. BourneUniversity of Virginia

Discussion

Loading...

Member takes

Implication

Key Points

Key points are not available for this paper at this time.

Cite This Study

Zhao et al. (2018) studied this question.

synapsesocial.com/papers/69db00961e19c8ae08835fcchttps://doi.org/10.1016/j.drudis.2018.01.035
View Full Paper
Ask AI
Bookmark
Share

Also Consider

Synapse has enriched 4 closely related papers on similar clinical questions. Consider them for comparative context:

  1. 1Kinetic and Catalytic Mechanisms of Protein Kinases2001 · 649 citations
  2. 2A Unique Structure for Epidermal Growth Factor Receptor Bound to GW572016 (Lapatinib)2004 · 1,135 citations
  3. 3Covalent Modifiers: A Chemical Perspective on the Reactivity of α,β-Unsaturated Carbonyls with Thiols via Hetero-Michael Addition Reactions2016 · 575 citations
  4. 4Genomic Determinants of PI3K Pathway Inhibitor Response in Cancer2012 · 98 citations