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October 2, 2006Angewandte Chemie International Edition264 citations

Oxetanes as Promising Modules in Drug Discovery

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GWGeorg WuitschikMRMark Rogers‐EvansKMKlaus Müller

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Abstract

Ring the changes: Introduction of an oxetane ring results in remarkably improved physico- and biochemical properties of the underlying scaffold. The oxetane ring confers enhanced solubility, reduces the metabolic degredation, lipophilicity, and amphiphilicity, and modulates the basicity of a nearby amine group.

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Wuitschik et al. (2006) studied this question.

synapsesocial.com/papers/6a639c861b4652261c6a8974https://doi.org/10.1002/anie.200602343
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