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October 7, 2015Journal of Cellular PhysiologyOpen Access

The Nox1/4 Dual Inhibitor GKT137831 or Nox4 Knockdown Inhibits Angiotensin‐II‐Induced Adult Mouse Cardiac Fibroblast Proliferation and Migration. AT1 Physically Associates With Nox4

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Key result

Nox4 knockdown, DPI, and the Nox1/4 dual inhibitor GKT137831 attenuated Angiotensin-II-induced mouse cardiac fibroblast proliferation and migration.

Why the study?

Does Nox4 inhibition or knockdown prevent Angiotensin-II-induced proliferation and migration in adult mouse cardiac fibroblasts?

Population

Adult mouse cardiac fibroblasts (CF)

Comparison

Nox4 knockdown, Nox inhibitor DPI, Nox1/Nox4… vs Control or Angiotensin-II alone

Design

Preclinical

Authors

NSNaveen K SomannaAVAnthony J. ValenteMKMaike Krenz

Discussion

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Overview

No immediate clinical implications for hypertensive heart disease; leaves open Nox4/IL-18 as mechanistic targets for further study.

Structured PICO

Does Nox4 inhibition or knockdown prevent Angiotensin-II-induced proliferation and migration in adult mouse cardiac fibroblasts?

P
Population
Adult mouse cardiac fibroblasts (CF)
I
Intervention
Nox4 knockdown, Nox inhibitor DPI, Nox1/Nox4 dual inhibitor GKT137831, IL-18 neutralization, MMP9 knockdown, or antioxidants (NAC, Tempol, MnTBAP, MnTMPyP)
C
Comparator
Control or Angiotensin-II alone
O
Outcome
Cardiac fibroblast proliferation and migrationsurrogate

Inhibition of Nox4 or the AT1/Nox4 interaction attenuates Angiotensin-II-induced cardiac fibroblast proliferation and migration, highlighting a potential therapeutic target for chronic hypertension-induced adverse cardiac remodeling.

Cite This Study

Somanna et al. (2015) studied Angiotensin-II-induced cardiac fibroblast proliferation and migration. Nox4 knockdown, DPI, or GKT137831 was evaluated on Cardiac fibroblast proliferation and migration. Nox4 knockdown, DPI, and the Nox1/4 dual inhibitor GKT137831 attenuated Angiotensin-II-induced mouse cardiac fibroblast proliferation and migration.

synapsesocial.com/papers/6a6ce78331a3df824326d87chttps://doi.org/10.1002/jcp.25210
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Also Consider

Synapse has enriched 3 closely related papers on similar clinical questions. Consider them for comparative context:

  1. 1Acetylsalicylic Acid Inhibits IL-18-Induced Cardiac Fibroblast Migration Through the Induction of RECK2013 · 39 citations
  2. 2Wnt-induced secreted protein-1 is a prohypertrophic and profibrotic growth factor2007 · 110 citations
  3. 3Nox4 Is a Protective Reactive Oxygen Species Generating Vascular NADPH Oxidase2012 · 623 citations