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October 20, 2020Trends in Pharmacological SciencesOpen Access

Critical Assessment of G Protein-Biased Agonism at the μ-Opioid Receptor

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Authors

AGAlexander GillisUNSW SydneyAKAndrea KliewerInsermEKEamonn KellyUniversity of Bristol

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Gillis et al. (2020) studied this question.

synapsesocial.com/papers/6a7161be75498292b70ada8ehttps://doi.org/10.1016/j.tips.2020.09.009
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  4. 4Mitragynine/Corynantheidine Pseudoindoxyls As Opioid Analgesics with Mu Agonism and Delta Antagonism, Which Do Not Recruit β-Arrestin-22016 · 328 citations