Why the study?
Do visnagin and diphenylurea prevent doxorubicin-induced cardiomyopathy in preclinical models?
Population
Zebrafish doxorubicin-induced cardiomyopathy model, cultured cardiomyocytes, mouse hearts, cultured tumor…
Comparison
Visnagin (VIS) and diphenylurea (DPU) vs Doxorubicin alone
Design
Preclinical
Authors
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Hypothesis-generating for MDH2 inhibition in doxorubicin cardiotoxicity; human trials needed before any clinical consideration.
Do visnagin and diphenylurea prevent doxorubicin-induced cardiomyopathy in preclinical models?
Visnagin and diphenylurea protect against doxorubicin-induced cardiotoxicity in preclinical models by modulating mitochondrial malate dehydrogenase (MDH2), without impairing anticancer efficacy.
Liu et al. (2014) studied this question.
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