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January 1, 2016BioMed Research InternationalOpen Access

Oral administration of AcSDKP, alone or with imidapril, ameliorated glomerulosclerosis and tubulointerstitial fibrosis and restored plasma cystatin C levels in diabetic mice.

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Why the study?

Does oral AcSDKP ameliorate kidney fibrosis in mouse models of diabetic nephropathy?

Population

Two mouse models of diabetic nephropathy: streptozotocin- induced type 1 diabetic CD-1 mice and type 2…

Comparison

Oral N-acetyl-seryl-aspartyl-lysyl-proline alone… vs Imidapril alone or untreated control

Design

Preclinical

Key result

Oral administration of AcSDKP, alone or with imidapril, ameliorated glomerulosclerosis and tubulointerstitial fibrosis and restored plasma cystatin C levels in diabetic mice.

Authors

KNKyoko NittaSSSen ShiTNTakako Nagai

Discussion

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Overview

Supports AcSDKP investigation in diabetic nephropathy; leaves open human translation and clinical utility.

Structured PICO

Does oral AcSDKP ameliorate kidney fibrosis in mouse models of diabetic nephropathy?

P
Population
Mouse models of type 1 and type 2 diabetic nephropathy.
I
Intervention
Oral N-acetyl-seryl-aspartyl-lysyl-proline (AcSDKP) alone or in combination with the ACE inhibitor imidapril
C
Comparator
Imidapril alone or untreated control
O
Outcome
Glomerulosclerosis and tubulointerstitial fibrosissurrogate

Oral administration of the endogenous peptide AcSDKP ameliorates kidney fibrosis and restores antifibrotic microRNAs in mouse models of type 1 and type 2 diabetic nephropathy.

Cite This Study

Nitta et al. (2016) studied Diabetic nephropathy. Oral AcSDKP vs. Imidapril alone or untreated was evaluated on Glomerulosclerosis, tubulointerstitial fibrosis, and plasma cystatin C levels. Oral administration of AcSDKP, alone or with imidapril, ameliorated glomerulosclerosis and tubulointerstitial fibrosis and restored plasma cystatin C levels in diabetic mice.

synapsesocial.com/papers/6a748ff480fadadbba0914e1https://doi.org/10.1155/2016/9172157
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Also Consider

Synapse has enriched 5 closely related papers on similar clinical questions. Consider them for comparative context:

  1. 1Renal Antifibrotic Effect of N-Acetyl-Seryl-Aspartyl-Lysyl-Proline in Diabetic Rats2013 · 30 citations
  2. 2Prevention of myocardial fibrosis by N-acetyl-seryl-aspartyl-lysyl-proline in diabetic rats2009 · 33 citations
  3. 3<i>N</i> -Acetyl-Seryl-Aspartyl-Lysyl-Proline Attenuates Renal Injury and Dysfunction in Hypertensive Rats With Reduced Renal Mass2009 · 47 citations
  4. 4N‐acetyl‐seryl‐aspartyl‐lysyl‐proline mediates the anti‐fibrotic properties of captopril in unilateral ureteric obstructed BALB/C mice2017 · 12 citations
  5. 5Antifibrotic effect of Ac-SDKP and angiotensin-converting enzyme inhibition in hypertension2004 · 97 citations