Direct Amination of Azoles via Catalytic C−H, N−H Coupling

Also Consider

Synapse has enriched 5 closely related papers on similar clinical questions. Consider them for comparative context:

1. 1Activated Aryl Chlorides: Useful Partners for the Coupling with 2‐Substituted Thiazoles in the Palladium‐Catalysed C‐H Activation/Functionalisation Reaction2007 · 68 citations
2. 2Intermolecular Amidation of Unactivated sp² and sp³ C−H Bonds via Palladium-Catalyzed Cascade C−H Activation/Nitrene Insertion2006 · 672 citations
3. 3Toward a Synthetically Useful Stereoselective C−H Amination of Hydrocarbons2007 · 381 citations
4. 4Palladium-catalyzed formation of carbon-nitrogen bonds. Reaction intermediates and catalyst improvements in the hetero cross-coupling of aryl halides and tin amides1994 · 845 citations
5. 5Synthesis of β-, γ-, and δ-Lactams via Pd(II)-Catalyzed C−H Activation Reactions2008 · 493 citations