Key result
Modulation of cGMP-PKG has entered clinical practice for pulmonary hypertension and erectile dysfunction, but translation to clinical success in heart failure has failed thus far.
Design
Review
Authors
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Cautions against premature PKG-based HF therapies; leaves open optimized translation strategies.
Understanding novel non-canonical roles of PKG1 is necessary for successful clinical translation of cGMP-PKG modulation therapies in heart failure.
Rainer et al. (2016) conducted a review in Heart failure and cardiovascular disease. cGMP-PKG modulation was evaluated. Modulation of cGMP-PKG has entered clinical practice for pulmonary hypertension and erectile dysfunction, but translation to clinical success in heart failure has failed thus far.
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