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June 1, 1994Nucleosides and Nucleotides

Synthesis and Antiviral Study of Dihydrothieno and Thianopyrimidine Diones Acyclic Nucleosides As Potential Anti-HIV Agents

Jacques Renault DANIEL LADUREE M. ROBBA

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Abstract

Acyclic nucleosides were prepared by alkylation of dihydrothieno and thianopyrimidines diones following Vorbruggen and Niedballa's method.(1) None of these HEPT analogues showed significant activity against Human Immunodeficiency Virus-1 (HIV-1)

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Renault et al. (1994) studied this question.

synapsesocial.com/papers/6a7e753355c19762e2b2a323 https://doi.org/10.1080/15257779408011884

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Synapse has enriched 5 closely related papers on similar clinical questions. Consider them for comparative context:

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