Key result
Procaine induces vasorelaxation in isolated rat aorta through multiple mechanisms, including nitric oxide release and activation of specific K+ channels.
Population
Isolated rat aortic rings
Comparison
Procaine (0.01-3 mM) vs Vehicle/control or various inhibitors
Design
Preclinical
Authors
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No immediate clinical implications from rat aortic data; leaves open human applicability pending translational studies.
Procaine induces vasorelaxation in rat aorta through multiple mechanisms, including nitric oxide release, activation of specific K+ channels, and direct inhibition of calcium mobilization.
Huang et al. (1999) studied this question. Procaine was evaluated on Vasorelaxation. Procaine induces vasorelaxation in isolated rat aorta through multiple mechanisms, including nitric oxide release and activation of specific K+ channels.
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